Publicacións en colaboración con investigadores/as de French Institute of Health and Medical Research (15)

2019

  1. Alternative retinoid X receptor (RXR) ligands

    Molecular and Cellular Endocrinology, Vol. 491

2017

  1. Reduced adiponectin expression after high-fat diet is associated with selective up-regulation of ALDH1A1 and further retinoic acid receptor signaling in adipose tissue

    FASEB Journal, Vol. 31, Núm. 1, pp. 203-211

  2. Structure-activity relationship study of vitamin D analogs with oxolane group in their side chain

    European Journal of Medicinal Chemistry, Vol. 134, pp. 86-96

2015

  1. Modulation of Retinoic Acid Receptor Subtypes by 5- and 8-Substituted (Naphthalen-2-yl)-based Arotinoids

    ChemMedChem, Vol. 10, Núm. 8, pp. 1378-1391

2012

  1. Retinoid receptors and therapeutic applications of RAR/RXR modulators

    Current Topics in Medicinal Chemistry, Vol. 12, Núm. 6, pp. 505-527

2011

  1. Epigenetic profiling of the antitumor natural product psammaplin A and its analogues

    Bioorganic and Medicinal Chemistry, Vol. 19, Núm. 12, pp. 3637-3649

  2. Total synthesis of the proposed structures of the DNA methyl transferase inhibitors peyssonenynes, and structural revision of peyssonenyne B

    Organic and Biomolecular Chemistry, Vol. 9, Núm. 20, pp. 6979-6987

2010

  1. A unique secondary-structure switch controls constitutive gene repression by retinoic acid receptor

    Nature Structural and Molecular Biology, Vol. 17, Núm. 7, pp. 801-807

2009

  1. C3 halogen and C8″ substituents on stilbene arotinoids modulate retinoic acid receptor subtype function

    ChemMedChem, Vol. 4, Núm. 10, pp. 1630-1640

  2. Modulating retinoid X receptor with a series of (E)-3-[4-hydroxy-3-(3- alkoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)phenyl]acrylic acids and their 4-alkoxy isomers

    Journal of Medicinal Chemistry, Vol. 52, Núm. 10, pp. 3150-3158

2008

  1. Caged agonist of P2Y1 and P2Y12 receptors for light-directed facilitation of platelet aggregation

    Biochemical Pharmacology, Vol. 75, Núm. 6, pp. 1341-1347

  2. Nuclear receptor ligand-binding domains: Reduction of helix H12 dynamics to favour crystallization

    Acta Crystallographica Section F: Structural Biology and Crystallization Communications, Vol. 64, Núm. 7, pp. 614-616

2007

  1. Design of selective nuclear receptor modulators: RAR and RXR as a case study

    Nature Reviews Drug Discovery, Vol. 6, Núm. 10, pp. 811-820

  2. Modulators of the structural dynamics of the retinoid X receptor to reveal receptor function

    Proceedings of the National Academy of Sciences of the United States of America, Vol. 104, Núm. 44, pp. 17323-17328

2005

  1. Characterization of the interaction between retinoic acid receptor/retinoid X receptor (RAR/RXR) heterodimers and transcriptional coactivators through structural and fluorescence anisotropy studies

    Journal of Biological Chemistry, Vol. 280, Núm. 2, pp. 1625-1633